"目錄號: HY-14390
LAS101057 是一種有效的周拐，選擇性的张咳，可口服的A2B receptor拮抗劑鼎俘。
相關(guān)產(chǎn)品
Preladenant-Vipadenant-CGS 21680 Hydrochloride-ZM241385-Istradefylline-Tozadenant-SCH 58261-Theophylline-Regadenoson-Capadenoson-IB-MECA-Ticlopidine hydrochloride-2-Cl-IB-MECA-N6-[2-(4-Aminophenyl)ethyl]adenosine-N6-Cyclohexyladenosine-
生物活性
Description
LAS101057 is a potent, selective, and orally efficaciousA2B receptorantagonist.
In Vivo
At 3 mg/kg, LAS101057 is active in preventing methacholine-induced AHR, and at 10 mg/kg it inhibits AHR to methacholine to a level virtually equal to that seen with dexamethasone at 1 mg/kg[1].
References
